Summaries of MND Research Institute-funded research programmes:

2010 Research Grants

In November 2009 the MND Research Institute of Australia approved grants to the following researchers to assist with their projects during 2010.  

Grants-in-aid

Grant-in-aid

Dr Julie Atkin    

Brain Injury & Repair Group, Howard Florey Institute, University of Melbourne

Is Protein Disulphide Isomerase (PDI) a novel biomarker for motor neuron disease?

There is currently no early diagnostic test for MND and usually lengthy and detailed clinical investigations are necessary.  The evidence we obtained in earlier studies has led us to believe that a protein called PDI may be a new and effective biomarker of MND.  In this study we will examine a large group of MND patients in comparison to unaffected individuals, to determine whether PDI could be used to reliably measure disease outcome and progression, and to predict disease in patients with inherited forms of MND.  If PDI can reliably diagnose MND, this would facilitate future studies to establish a diagnostic kit for MND or to design clinical trials of new drugs.

 

 

Peter Stearne Grant for Familial MND

Dr Ian Blair

Northcott Laboratory, ANZAC Research Institute, NSW. 

Characterisation and investigation of a new transgenic mouse model expressing mutant TDP-43.

The only proven causes of MND are mutations in genes that lead to death of motor neurons.  Using these mutations, mice have previously been developed that mimic features of MND.  These animals, called mouse models of MND, have been a principal tool for testing proposed disease treatments. Unfortunately the promise of treatments shown in existing mouse models have largely proven unsuccessful in human trials. We recently described mutations in a new MND gene, TDP-43.  We have developed a new mouse that carries one of these TDP-43 mutations.  We now aim to monitor and test this mouse to establish whether it develops similar symptoms to MND.  If so, this new mouse model will be available for investigating the biology of the disease and for evaluating treatments.

 

 

Mick Rodger MND Research Grant

A/Prof Meng Inn Chuah

Menzies Research Institute, University of Tasmania

Effect of metallothionein and exercise on progression of motor neurone disease.

Amyotrophic lateral sclerosis (ALS) is the major cause of motor neurone diseases (MND), which are progressive and ultimately fatal diseases caused by the degeneration of motor neurons in the brain and spinal cord of patients.  Unfortunately there are no effective clinical treatments available that can protect motor neurones from such death, with the only drug currently available, riluzole (rilutek) conferring only a very modest alleviation in symptoms, and is only effective over a short period of several months.  Metallothionein (MT) proteins are known to be powerfully neuroprotective in several experimental models of neuronal injury and disease including ALS.  We now have preliminary data suggesting that administration of MT might be effective in prolonging survival in an animal model of ALS. This project will explore further this therapeutic potential by assessing the possible benefits of combining MT with an exercise regimen to improve the functional and survival outcome of a mouse model of ALS.

 

Grant-in-aid

Dr Peter Crouch

Dept of Pathology, University of Melbourne, VIC

Investigating cellular hypoxia as a causative factor in MND and as a potential therapeutic target.

The fundamental biological causes of decreased motor neurone function in MND remain unknown.  Genetic clues are evident in familial forms of the disease, but familial MND only accounts for a small minority of all cases and these genetic clues therefore cannot explain the majority of cases. Identifying the causes decreased motor neurone function is an essential step in developing new and more effective therapeutics to treat MND.  The research described in this application focuses on demonstrating the mechanism of action for a novel therapeutic compound shown to be effective in MND model mice. Undertaking the described work presents a unique opportunity to simultaneously progress the development of this compound towards clinical trials, and to identify what may be an important biological contributor to all forms of MND.

Our work to date has shown that the copper-based compound CuII(atsm) significantly delays the onset of MND-like symptoms in a mouse model of the disease.  Most importantly, CuII(atsm) delays the onset of paralysis in these mice. Parallel work has started to reveal important information on how CuII(atsm) may mediate its therapeutic effects.  Essentially, we have shown that CuII(atsm) is a relatively inert compound, but when exposed to cells grown with inadequate oxygen supply, the CuII(atsm) becomes activated. When activated, CuII(atsm) induces cellular responses that have the potential to improve neuronal function.  This work is highly significant when considered in the context of current MND research, as emerging evidence indicates that impaired cellular responses to inadequate oxygen supply can induce development of MND.

The research described in this application will provide information on the cellular conditions that induce activation of CuII(atsm) and therefore generate its therapeutic activity in MND model mice.  In addition, it will provide new information on cellular responses to oxygen supply as a potential biological cause of MND.

 

 

Zo-eč MND Research Grant

Dr Fiona Fisher

Neuropsychology, Calvary Health Care Bethlehem, VIC

Emotion recognition and social communication in MND: impact on behaviour and carer burden.

In recent years, there has been a surge of research into the non-motor symptoms of MND, with the impact of MND on thinking skills, behaviour and emotional functioning being more widely accepted. Research, while limited at this stage, has shown that MND can damage parts of the brain that are essential for normal understanding of emotions, and in particular in understanding the non-verbal aspects of communication that indicate the emotional states of others. What this means is that some people with MND may have trouble with the finer, more subtle details of social communication, social cognition and the ability behave appropriately in their social interactions with other people.  These emotional processing changes have the potential to impact upon the relationship between persons with MND and their carers.

The proposed research project aims to investigate previously identified social-emotional changes and investigate the relationship of such changes with alterations in behaviour. In addition, the relationship between social-emotions difficulties and carer burden will be explored. This will provide new information about the frequency and impact of emotional processing difficulties in people with MND. It will also increase understanding of the relationship of such difficulties to social communication, behavioural changes and carer burden.

 

 

Grant-in-aid

Dr Robert Henderson

Dept of Neurology, Royal Brisbane and Women's Hospital, QLD

Novel markers of motor neurone disease- quantitative upper and lower motor neurone markers.

Motor Neurone Disease (MND) is a relentlessly progressive disorder of upper and lower motor neurones.  Since the first description of MND in the 19th century, only one drug (riluzole) with modest disease-modifying potency has been developed. The diagnosis of this disorder is clinical and there is a significant delay between the symptom onset and diagnosis, possibly beyond the therapeutic window.  Clinical signs and functional scales are inadequate for detection or quantification of the loss of upper and lower motor neurones. That is the reason why patient survival has been the measure of therapeutic response in many trials. However, the heterogeneity in the rate of progression and survival in MND patients is challenging the outcome of clinical trials.

Our research project focuses on novel markers that are sensitive to the progression of disease, which might enhance the diagnostic algorithm and might be useful to monitor the effectiveness of new therapies.  We perform neuroimaging and neurophysiology studies to identify objective upper and lower neurone markers. In combination, these quantitative markers might be sensitive to early therapeutic effects and might also resolve complexities of phenotypic heterogeneity in clinical trials.

Hence, we evaluate longitudinally patients with different clinical phenotypes of MND (e.g. UMN or LMN predominant, pure LMN type) to quantify the rate of progression and to understand if the degeneration of the upper and lower segments is simultaneous, or if independent that neither is the cause or the consequence of the other.

 

 

Grant-in-aid

Dr Qiao-Xin Li

Dept of Pathology, University of Melbourne, VIC

Investigating the in vivo targets affected by a novel therapeutic agent for motor neuron disease.

Motor Neuron Disease (MND) affects the motor system required to maintain muscle control.  Inevitably the disease progresses to paralysis and premature death, within 3-5 years after diagnosis.  There are limited therapeutic options available for treating the disease.  Our current work has identified a compound, known as CuII(atsm), that substantially delays the development of disease symptoms in a mouse model of MND.  This proposal is to investigate the optimal treatment scheme for the CuII(atsm) before advancing to preclinical trials, as well as the identification of in vivo targets of CuII(atsm). Ultimately this study will help expedite the development of effective MND therapeutic strategies.

 

 

Grant-in-aid

Dr Hakan Muyderman

Medical Biochemistry & Human Physiology, Flinders University, SA

The role of TDP-43 in astrocytes in motor neuron disease.

The presence of cellular inclusion bodies links a large spectrum of neurological diseases together, including motor neuron disease (MND). Recently, the TAR-DNA-binding protein TDP-43 was identified as a primary component of these inclusions and mutations in the gene encoding for this protein have been causally linked to familiar forms of MND. However TDP-43 positive inclusions are not only present in motor neurons but also in surrounding glial cells, predominately in astrocytes. Although there is no loss of these cells in MND, affected astrocytes have pronounced changes in expression of genes regulating essential cellular functions. In addition, in some models of MND, sick astrocytes kill healthy motor neurons when the two cell types are grown in culture. Based on these and similar data it has been suggested that motor neuron cell death could partly result from deficiencies in the interaction between motor neurons and astrocytes. However the role of TDP-43 in the interplay between these two cell types is not known.

 

In this context, results recently obtained in our laboratory demonstrate that astrocytes expressing TDP-43 mutations also suffer from changes in normal cell function. Moreover, several of these changes have the potential to severely affect function and survival of motor neurons. Based on these results, we hypothesise that astrocytes expressing human TDP-43 mutations will impair normal motor neuron function and survival. This hypothesis, which has not been tested, constitutes the overall aim of this project. We believe that a successful identification of astrocytic TDP-43 protein as a component in the pathology of motor neuron disease will present new targets for therapeutic interventions where none exists and will aid in understanding a range of related neurodegenerative diseases.

 

 

Grant-in-aid

A/Prof Roger Pamphlett

Stacey MND Laboratory, University of Sydney

Looking for abnormal gene expression in ALS spinal cords using next-generation sequencing.

  • Most researchers now believe that genetic abnormalities underlie sporadic ALS (SALS). Increasing evidence suggests RNA metabolism may be abnormal in ALS.

  • A powerful way to uncover genetic abnormalities underlying a disease is to extract RNA from the tissue most affected by the disease, and see if this differs from normal tissue.

  • RNA can be abnormal in being (1) under-expressed, (2) over-expressed, or (3) of an abnormal type (e.g., a product with a “misspelling” or an unusual composition of exons).

  • Until now, technological limitations have restricted the use of measuring RNA gene expression to a relatively small number of genes.

  • The latest next-generation sequencing methods can now examine all the RNA transcripts from the entire human genome.

  • We will use Illumina next-generation high-throughput sequencing to examine the complete RNA expression within SALS spinal cords.

  • This study will give us the most complete picture to date of gene behaviour in SALS.

  • These findings will have a direct bearing on any future gene therapy in SALS.

 

Grant-in-aid

Dr Mary-Louise Rogers & Prof Robert Rush

Dept of Human Physiology, Flinders University SA

A bio-marker for motor neurone disease.

Diagnosis of motor neurone disease is usually a long, drawn out process that creates anxiety for patients and their families. We are working to find a bio-molecule in urine that can be used to easily diagnose motor neurone disease. This 'biomarker' of the disease will be valuable as a way of objectively measuring progression of the disease and also for determining whether new drugs have value in the treatment of this devastating illness.

 

 

Grant-in-aid

Dr Bradley Turner  

Florey Neuroscience Institutes, University of Melbourne

A role for survival motor neuron protein in MND?

Understanding the earliest and central pathological events in MND is essential to developing effective treatments. We recently showed that survival motor neuron (SMN) protein levels are lower in laboratory models of MND. SMN deficiency occurs very early before motor neuron loss and symptoms in MND model mice, suggesting that it may be an important mechanism for disease.  We now wish to determine whether MND patients are deficient in SMN and whether this correlates with age of diagnosis and disease severity. These studies will indicate whether SMN replacement may be considered useful for MND therapy.

 

 

Charles & Shirley Graham MND Research Grant

Dr Robyn Wallace

Queensland Brain Institute

Identifying genes that are affected by MND causing TDP-43 mutations.

Protein tangles that aggregate in affected nerve cells are a pathological hallmark of MND.  Recent studies have demonstrated that TAR DNA-binding protein (TDP-43) is a principal component of these nerve cell aggregates.  This was a major breakthrough in the understanding of MND.  However, the function of TDP-43 in the nervous system is currently unknown and its role in the pathogenesis of MND remains unclear. Genetic mutations associated with both familial and sporadic MND have recently been identified in TDP-43.  These mutations offer a unique opportunity to determine how abnormal TDP-43 leads to loss of motor neurons in MND patients.  The aim of this project is to investigate how these mutations affect the normal function of TDP-43.  Specifically, we will identify genes that are regulated by TDP-43 and determine whether these genes are altered in MND patients with TDP-43 mutations.  These studies will improve our understanding of what causes MND and provide rational targets for new therapies.

 

 

Mick Rodger Benalla MND Research Grant

Dr Anthony White

Dept of Pathology, University of Melbourne, VIC

Investigating the role of biometals in abnormal metabolism of TDP-43.

Motor neuron disease is a devastating and rapidly progressing illness affecting adults and often results in death within 2-5 years of diagnosis.  No effective treatments or cure exists.  Despite extensive research into the underlying causes of motor neuron cell death, the processes are still poorly understood.  Recent discoveries have identified a protein thought to have a key role in the pathways leading to motor neuron degeneration.  This protein, TDP-43, had been shown to undergo fragmentation into smaller pieces (called C-terminal fragments, CTFs), followed by aggregation into clumps and are also modified by phosphorylation and ubiquitination.  This process is believed to be associated with motor neuron degeneration. However, little is known of the key early processes that lead to TDP-43 fragmentation and aggregation or how this results in motor neuron cell death.  We have developed a cell culture model based on use of a motor neuron cell line to investigate factors that influence disease-associated changes to TDP-43.  We have so far found that zinc (an important biometal in the brain and neurodegeneration) can induce specific TDP-43 aggregation.  We are now further investigating this novel finding and using a unique protein array-based approach to map molecular pathways of TDP-43-mediated motor neuron cell death.  The outcomes of this project will provide a significant advance in our understanding of TDP-43 in motor neuron disease and may lead to development of novel treatment approaches for patients with the disease.

 

 

Bill Gole Postdoctoral Fellowship for MND Research 2010 - 2012

Dr Shu Yang

Northcott Laboratory, ANZAC Research Institute, NSW. 

Investigating the role of recently identified mutant genes in MND pathogenesis.

The disease mechanism underlying motor neuron disease (MND) is currently poorly understood, making the development of diagnostic tools and therapeutics difficult.  However, proteins that play fundamental roles in MND pathogenesis have recently been identified, providing new hope for understanding the cause of MND and development of therapeutic and diagnostic tools.  The 43 kDa TAR DNA binding protein (TDP-43) was recently identified as a signature component of the abnormal protein aggregates found in the brain and spinal cord of most sporadic and familial MND patients.  Our group identified several mutant forms of TDP-43 that appear to directly trigger neurodegeneration leading to MND (funded by a Bill Gole Fellowship to Dr Blair, 2006-2007).  We hypothesise that identifying the mechanisms through which rare TDP-43 mutations cause MND will be more widely relevant to understanding the cause of familial and sporadic MND.  We will establish novel TDP-43-expressing MND cell models and a transgenic mouse model to study the function of mutant TDP-43 protein. 

The significance of the proposed project includes a greater understanding of how mutant TDP-43 leads to protein aggregation and motor neuron degeneration in MND, as well as knowledge of the functions of other signature proteins in MND, such as FUS, that may provide new diagnostic and therapeutic targets.  The establishment of the TDP-43 transgenic mouse model may provide a better model to understand sporadic MND pathogenesis than the existing SOD1 transgenic mouse models. This model may also act as a useful platform for MND therapeutic development.

 

 

Grants awarded in previous years continue in 2010 for:

Dr James Burrell

Prince of Wales Medical Research Institute, NSW.

PhD Scholarship for MND Research 2009 - 2011, co-funded with NHMRC

Cognition and behaviour in motor neuron disease.

Motor neuron disease (MND) and fronto-temporal dementia (FTD) are fatal neurodegenerative disorders of unknown cause. There are poorly understood clinical and pathological overlaps between MND and FTD which this research aims to clarify. The impact of cognitive deficits on carer burden will also be investigated. It is hoped that this research may contribute to the development of a pathological model that explains the development of MND and FTD.

 

 

Dr Justin Yerbury  

Centre for Medical Biosciences, University of Wollongong

Bill Gole Postdoctoral Fellowship for MND Research 2009 - 2011

Probing molecular mechanisms of microglial and astrocyte activation in ALS.

This project combines unique expertise to perform truly pioneering studies to determine how a genetic defect in a protein, superoxide dismutase, affects immune processes implicated in motor neuron disease. Novel approaches will be used to study relevant molecular interactions, both in the test tube and in animal models. The outcomes will provide a new understanding of these processes and may contribute towards the ultimate development of new therapies.

 

Recent research suggests that a soluble factor in ALS CSF is toxic to motor neurones via both direct and indirect effects; the latter is thought to involve activation of microglial cells which secrete toxic mediators.  One potential soluble factor that may promote cell activation and neurotoxicity is extracellular mSOD1.    This project will provide significant insights into the mechanisms by which extracellular mSOD1 influences the development of familial ALS (fALS) pathology. We expect that the research outcomes will stimulate a high level of general interest resulting in publications in high impact international scientific journals and provide vital clues to possible new directions for therapies to combat fALS, for which there is currently no effective treatment.

 

 

Dr Anna King

NeuroRepair Group, Menzies Research Institute, University of Tasmania.

Bill Gole Postdoctoral Fellowship for MND Research 2008 - 2010

Investigating the causes and consequence of axonal pathology in amyotrophic lateral sclerosis.

Motor neuron disease (MND) is caused by a loss of function of the nerve cells controlling the muscles. I have recently developed a cell culture model which mimics the degenerative changes in motor nerve cells that underlie the onset of amyotrophic lateral sclerosis, the major cause of human MND.  I will use this model to investigate the factors and mechanisms that cause motor neurons to degenerate, an approach which may indicate new therapeutic opportunities for an otherwise incurable condition.

 

 

Dr Jennica Winhammar

The Prince of Wales Medical Research Institute, NSW.

Bill Gole Postdoctoral Fellowship for MND Research 2008 - 2010

Clinical trial to assess the neuroprotective properties of a sodium channel blocking agent in motor neurone disease.

 This project will provide clinical trial information related to the potential neuroprotective properties of a sodium channel blocking agent in patients with motor neurone disease. Specifically, it will establish whether the sodium channel blocking agent can slow disease progression.  A potential therapeutic response would provide impetus for a larger scale, multi-centre clinical trial. In addition to providing information about potential mechanisms of neurodegeneration and their treatment, new quantifiable measures will be further developed to objectively monitor MND patients in a clinical trials setting.

 

 

 

Funding over three years is also being provided for the MND Research Tissue Bank of Victoria (2008 - 2010)